Matches in SemOpenAlex for { <https://semopenalex.org/work/W1993791556> ?p ?o ?g. }
- W1993791556 endingPage "1666" @default.
- W1993791556 startingPage "1651" @default.
- W1993791556 abstract "After 7 years from its cloning, the transient receptor potential vanilloid type-1 (TRPV1) channel remains the sole membrane receptor mediating the pharmacological effects of the hot chilli pepper pungent component, capsaicin, and of the Euphorbia toxin, resiniferatoxin. Yet, this ion channel represents one of the most complex examples of how the activity of a protein can be regulated. Among the several chemicophysical stimuli that can modulate TRPV1 permeability to cations, endogenous lipids appear to play a major role, either as allosteric effectors or as direct agonists, or both. Furthermore, the capability of some mediators, such as the endocannabinoid anandamide, or the eicosanoid precursors 12- and 5-hydroperoxy-eicosatetraenoic acids, to activate TRPV1 receptors provides a striking example of the site-dependent and metabolic functional plasticity, respectively, typical of bioactive lipids. In this article, the multi-faceted and most recently discovered aspects of TRPV1 regulation are reviewed, with particular emphasis on the interaction between these membrane channels and some lipid molecules." @default.
- W1993791556 created "2016-06-24" @default.
- W1993791556 creator A5007484138 @default.
- W1993791556 creator A5076395210 @default.
- W1993791556 date "2005-08-01" @default.
- W1993791556 modified "2023-09-27" @default.
- W1993791556 title "Lipids as regulators of the activity of transient receptor potential type V1 (TRPV1) channels" @default.
- W1993791556 cites W1488329806 @default.
- W1993791556 cites W1492591187 @default.
- W1993791556 cites W1495409864 @default.
- W1993791556 cites W1511198581 @default.
- W1993791556 cites W1564453175 @default.
- W1993791556 cites W1569255175 @default.
- W1993791556 cites W1570505030 @default.
- W1993791556 cites W1571969265 @default.
- W1993791556 cites W1638666422 @default.
- W1993791556 cites W1883732752 @default.
- W1993791556 cites W1901115344 @default.
- W1993791556 cites W1923600385 @default.
- W1993791556 cites W1964358846 @default.
- W1993791556 cites W1966440880 @default.
- W1993791556 cites W1968366571 @default.
- W1993791556 cites W1969338731 @default.
- W1993791556 cites W1971566600 @default.
- W1993791556 cites W1971754431 @default.
- W1993791556 cites W1973528953 @default.
- W1993791556 cites W1979608920 @default.
- W1993791556 cites W1981377088 @default.
- W1993791556 cites W1984033377 @default.
- W1993791556 cites W1985030046 @default.
- W1993791556 cites W1986235007 @default.
- W1993791556 cites W1986263012 @default.
- W1993791556 cites W1988375390 @default.
- W1993791556 cites W1988531294 @default.
- W1993791556 cites W1991050464 @default.
- W1993791556 cites W1992001407 @default.
- W1993791556 cites W1992358268 @default.
- W1993791556 cites W1993476176 @default.
- W1993791556 cites W1993763215 @default.
- W1993791556 cites W1995705528 @default.
- W1993791556 cites W1997308301 @default.
- W1993791556 cites W1998612393 @default.
- W1993791556 cites W1998698456 @default.
- W1993791556 cites W1999667297 @default.
- W1993791556 cites W2005828463 @default.
- W1993791556 cites W2006383469 @default.
- W1993791556 cites W2009326432 @default.
- W1993791556 cites W2010665440 @default.
- W1993791556 cites W2016034906 @default.
- W1993791556 cites W2016164238 @default.
- W1993791556 cites W2017047663 @default.
- W1993791556 cites W2019969188 @default.
- W1993791556 cites W2020352730 @default.
- W1993791556 cites W2020414448 @default.
- W1993791556 cites W2021138861 @default.
- W1993791556 cites W2021815265 @default.
- W1993791556 cites W2021876302 @default.
- W1993791556 cites W2022819833 @default.
- W1993791556 cites W2023486326 @default.
- W1993791556 cites W2024122340 @default.
- W1993791556 cites W2027256301 @default.
- W1993791556 cites W2029993965 @default.
- W1993791556 cites W2030894292 @default.
- W1993791556 cites W2040044089 @default.
- W1993791556 cites W2040664792 @default.
- W1993791556 cites W2041743176 @default.
- W1993791556 cites W2043033522 @default.
- W1993791556 cites W2043271992 @default.
- W1993791556 cites W2045626430 @default.
- W1993791556 cites W2049100687 @default.
- W1993791556 cites W2049727782 @default.
- W1993791556 cites W2050346904 @default.
- W1993791556 cites W2052214708 @default.
- W1993791556 cites W2054154138 @default.
- W1993791556 cites W2056416370 @default.
- W1993791556 cites W2057039966 @default.
- W1993791556 cites W2057468498 @default.
- W1993791556 cites W2059742450 @default.
- W1993791556 cites W2062606765 @default.
- W1993791556 cites W2062713583 @default.
- W1993791556 cites W2063102563 @default.
- W1993791556 cites W2069460649 @default.
- W1993791556 cites W2071823593 @default.
- W1993791556 cites W2079108672 @default.
- W1993791556 cites W2081044920 @default.
- W1993791556 cites W2082947615 @default.
- W1993791556 cites W2083350393 @default.
- W1993791556 cites W2083484726 @default.
- W1993791556 cites W2085802434 @default.
- W1993791556 cites W2086881537 @default.
- W1993791556 cites W2087674201 @default.
- W1993791556 cites W2088511433 @default.
- W1993791556 cites W2088764206 @default.
- W1993791556 cites W2089956060 @default.
- W1993791556 cites W2090617423 @default.
- W1993791556 cites W2098443650 @default.
- W1993791556 cites W2100585655 @default.
- W1993791556 cites W2100713606 @default.