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- W1994421160 abstract "Aniracetam (1-p-anisoyl-2-pyrrolidinone) selectively reverses the anticonvulsant activities of the non-NMDA receptor antagonists, GYKI 52466 (1-4-aminophenyl)-4-methyl-7,8-methylenedioxy-5H-2,3-benzodiazepine · HCl) and, to a lesser extent, NBQX (2,3-dihydroxy-6-nitro-7-sulfamoylbenzo(F)quinoxaline), without affecting the anticonvulsant activity of the competitive NMDA receptor antagonist, D(−)-CPPene, in DBA/2 mice. Pretreatment with aniracetam (50 nmol i.c.v., 15 min before drugs) increases the ED50 values (μmol/kg i.p., 15 min) for GYKI 52466-induced protection against sound-induced clonic seizures in DBA/2 mice 7 fold, from 20.1 (11.9–33.9) to 142 (91.7–219), and for NBQX-induced protection 2 fold, from 39.7 (33.8–46.7) to 85.6 (63.9–115), respectively. Aniracetam on its own (12.5–100 nmol i.c.v.) has no convulsant activity, but reverses the anticonvulsant effect of GYKI 52466 (60 μmol/kg i.p., 15 min) in a dose-dependent manner." @default.
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- W1994421160 title "Aniracetam reverses the anticonvulsant action of NBQX and GYKI 52466 in DBA/2 mice" @default.
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- W1994421160 doi "https://doi.org/10.1016/0014-2999(93)90465-t" @default.
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