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- W1994869675 endingPage "4171" @default.
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- W1994869675 abstract "The potential use of antisense and siRNA oligonucleotides as therapeutic agents has elicited a great deal of interest. However, a major issue for oligonucleotide-based therapeutics involves effective intracellular delivery of the active molecules. In this Survey and Summary, we review recent reports on delivery strategies, including conjugates of oligonucleotides with various ligands, as well as use of nanocarrier approaches. These are discussed in the context of intracellular trafficking pathways and issues regarding in vivo biodistribution of molecules and nanoparticles. Molecular-sized chemical conjugates and supramolecular nanocarriers each display advantages and disadvantages in terms of effective and nontoxic delivery. Thus, choice of an optimal delivery modality will likely depend on the therapeutic context." @default.
- W1994869675 created "2016-06-24" @default.
- W1994869675 creator A5020122857 @default.
- W1994869675 creator A5040221227 @default.
- W1994869675 creator A5044182015 @default.
- W1994869675 creator A5083780909 @default.
- W1994869675 date "2008-05-23" @default.
- W1994869675 modified "2023-10-17" @default.
- W1994869675 title "Mechanisms and strategies for effective delivery of antisense and siRNA oligonucleotides" @default.
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