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- W1994927708 abstract "A galactoside prodrug has been designed that can be selectively activated by lysosomal β-galactosidase located inside cancer cells expressing a specific tumor-associated receptor. In their Communication on page 11606 ff. S. Papot and co-workers show that this efficient enzymatic process triggers a potent cytotoxic effect, releasing the potent antimitotic agent MMAE and allowing the destruction of both receptor-positive and surrounding receptor-negative tumor cells." @default.
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- W1994927708 date "2012-10-12" @default.
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- W1994927708 title "Inside Cover: The First Generation of β-Galactosidase-Responsive Prodrugs Designed for the Selective Treatment of Solid Tumors in Prodrug Monotherapy (Angew. Chem. Int. Ed. 46/2012)" @default.
- W1994927708 doi "https://doi.org/10.1002/anie.201207805" @default.
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