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- W1996039215 abstract "A series of 3-urea-1-(phenylmethyl)-pyridones was discovered as novel EP(3) antagonists via high-throughput screening and subsequent optimization. The synthesis, structure-activity relationships, and optimization of the initial hit that resulted in potent and selective EP(3) receptor antagonists such as 11g are described." @default.
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- W1996039215 date "2010-11-01" @default.
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- W1996039215 title "3-Urea-1-(phenylmethyl)-pyridones as novel, potent, and selective EP3 receptor antagonists" @default.
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- W1996039215 doi "https://doi.org/10.1016/j.bmcl.2010.08.137" @default.
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