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- W1996947378 endingPage "1266" @default.
- W1996947378 startingPage "1261" @default.
- W1996947378 abstract "G-protein-coupled receptor 40 (GPR40), known as free fatty acid receptor 1, is mainly expressed in pancreatic β-cells and activated by medium- and long-chain fatty acids. Increasing evidence indicates that the activation of GPR40 in cells causes insulin secretion, and GPR40 has become an attractive therapeutic target for type 2 diabetes. Recently, certain novel GPR40 agonists have been identified that regulate glucose-stimulated insulin secretion, leading to the development of new drugs for the treatment of type 2 diabetes. In this review, we focus on progress in the physiological role of GPR40 and potential drugs targeting GPR40 over the past decade." @default.
- W1996947378 created "2016-06-24" @default.
- W1996947378 creator A5011365911 @default.
- W1996947378 creator A5012363939 @default.
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- W1996947378 creator A5026071264 @default.
- W1996947378 creator A5039651131 @default.
- W1996947378 creator A5074051847 @default.
- W1996947378 date "2012-09-26" @default.
- W1996947378 modified "2023-10-03" @default.
- W1996947378 title "GPR40: A therapeutic target for mediating insulin secretion" @default.
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