Matches in SemOpenAlex for { <https://semopenalex.org/work/W1999477823> ?p ?o ?g. }
- W1999477823 endingPage "495" @default.
- W1999477823 startingPage "492" @default.
- W1999477823 abstract "We herein describe the systematic approach used to develop new analogues of compound 2, recently identified as a potent and selective fatty acid amide hydrolase (FAAH) inhibitor. Aiming at identifying new scaffolds endowed with improved drug disposition properties with respect to the phenylpyrrole-based lead, we subjected it to two different structural modification strategies. This process allowed the identification of derivatives 4b and 5c as potent, reversible and non-competitive FAAH inhibitors." @default.
- W1999477823 created "2016-06-24" @default.
- W1999477823 creator A5004950855 @default.
- W1999477823 creator A5006864475 @default.
- W1999477823 creator A5015069863 @default.
- W1999477823 creator A5023892631 @default.
- W1999477823 creator A5043670620 @default.
- W1999477823 creator A5045385809 @default.
- W1999477823 creator A5045815002 @default.
- W1999477823 creator A5060025183 @default.
- W1999477823 creator A5071576099 @default.
- W1999477823 creator A5073541643 @default.
- W1999477823 creator A5079124576 @default.
- W1999477823 creator A5081951082 @default.
- W1999477823 creator A5084489352 @default.
- W1999477823 creator A5084867757 @default.
- W1999477823 date "2013-01-01" @default.
- W1999477823 modified "2023-10-17" @default.
- W1999477823 title "Identification of a novel arylpiperazine scaffold for fatty acid amide hydrolase inhibition with improved drug disposition properties" @default.
- W1999477823 cites W1968933287 @default.
- W1999477823 cites W1998465336 @default.
- W1999477823 cites W2007924093 @default.
- W1999477823 cites W2008818829 @default.
- W1999477823 cites W2014306399 @default.
- W1999477823 cites W2018780060 @default.
- W1999477823 cites W2021843784 @default.
- W1999477823 cites W2027991357 @default.
- W1999477823 cites W2043896152 @default.
- W1999477823 cites W2044344430 @default.
- W1999477823 cites W2050752896 @default.
- W1999477823 cites W2079776672 @default.
- W1999477823 cites W2081573540 @default.
- W1999477823 cites W2085488617 @default.
- W1999477823 cites W2106462471 @default.
- W1999477823 cites W2128615732 @default.
- W1999477823 cites W2134623848 @default.
- W1999477823 cites W2136815394 @default.
- W1999477823 cites W2143544679 @default.
- W1999477823 cites W2160291493 @default.
- W1999477823 cites W2952078105 @default.
- W1999477823 cites W97923480 @default.
- W1999477823 doi "https://doi.org/10.1016/j.bmcl.2012.11.035" @default.
- W1999477823 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/23237837" @default.
- W1999477823 hasPublicationYear "2013" @default.
- W1999477823 type Work @default.
- W1999477823 sameAs 1999477823 @default.
- W1999477823 citedByCount "16" @default.
- W1999477823 countsByYear W19994778232013 @default.
- W1999477823 countsByYear W19994778232015 @default.
- W1999477823 countsByYear W19994778232016 @default.
- W1999477823 countsByYear W19994778232018 @default.
- W1999477823 countsByYear W19994778232019 @default.
- W1999477823 countsByYear W19994778232020 @default.
- W1999477823 countsByYear W19994778232021 @default.
- W1999477823 countsByYear W19994778232022 @default.
- W1999477823 countsByYear W19994778232023 @default.
- W1999477823 crossrefType "journal-article" @default.
- W1999477823 hasAuthorship W1999477823A5004950855 @default.
- W1999477823 hasAuthorship W1999477823A5006864475 @default.
- W1999477823 hasAuthorship W1999477823A5015069863 @default.
- W1999477823 hasAuthorship W1999477823A5023892631 @default.
- W1999477823 hasAuthorship W1999477823A5043670620 @default.
- W1999477823 hasAuthorship W1999477823A5045385809 @default.
- W1999477823 hasAuthorship W1999477823A5045815002 @default.
- W1999477823 hasAuthorship W1999477823A5060025183 @default.
- W1999477823 hasAuthorship W1999477823A5071576099 @default.
- W1999477823 hasAuthorship W1999477823A5073541643 @default.
- W1999477823 hasAuthorship W1999477823A5079124576 @default.
- W1999477823 hasAuthorship W1999477823A5081951082 @default.
- W1999477823 hasAuthorship W1999477823A5084489352 @default.
- W1999477823 hasAuthorship W1999477823A5084867757 @default.
- W1999477823 hasBestOaLocation W19994778232 @default.
- W1999477823 hasConcept C116834253 @default.
- W1999477823 hasConcept C148001335 @default.
- W1999477823 hasConcept C15744967 @default.
- W1999477823 hasConcept C170493617 @default.
- W1999477823 hasConcept C181199279 @default.
- W1999477823 hasConcept C185592680 @default.
- W1999477823 hasConcept C202751555 @default.
- W1999477823 hasConcept C21951064 @default.
- W1999477823 hasConcept C2776885963 @default.
- W1999477823 hasConcept C2777752112 @default.
- W1999477823 hasConcept C2778439535 @default.
- W1999477823 hasConcept C2780035454 @default.
- W1999477823 hasConcept C2780120296 @default.
- W1999477823 hasConcept C2781144285 @default.
- W1999477823 hasConcept C38022665 @default.
- W1999477823 hasConcept C543025807 @default.
- W1999477823 hasConcept C55493867 @default.
- W1999477823 hasConcept C59822182 @default.
- W1999477823 hasConcept C71240020 @default.
- W1999477823 hasConcept C71924100 @default.
- W1999477823 hasConcept C74187038 @default.
- W1999477823 hasConcept C77805123 @default.
- W1999477823 hasConcept C86803240 @default.
- W1999477823 hasConcept C98274493 @default.
- W1999477823 hasConceptScore W1999477823C116834253 @default.
- W1999477823 hasConceptScore W1999477823C148001335 @default.