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Matches in SemOpenAlex for { <https://semopenalex.org/work/W2000340739> ?p ?o ?g. }

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• W2000340739 abstract "The synthesis of imidazolidin-4-one derivatives of primaquine containing the five-membered ring at the C-terminus of a dipeptide backbone coupled to the parent drug is described. These peptidomimetic derivatives were active against a chloroquine-resistant Plasmodium falciparum strain and inhibited the development of the sporogonic cycle of Plasmodium berghei, affecting the appearance of oocysts in the midguts of the mosquitoes. The novel imidazolidin-4-ones are extremely stable, both in human plasma and in pH 7.4 buffer, as a result of N1-acylation. Thus, ‘internal’ imidazolidin-4-ones derived from dipeptidyl 8-aminoquinolines represent a new entry in antimalarial structure–activity relationships." @default.
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• W2000340739 date "2008-07-01" @default.
• W2000340739 modified "2023-09-23" @default.
• W2000340739 title "Imidazolidin-4-one peptidomimetic derivatives of primaquine: Synthesis and antimalarial activity" @default.
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• W2000340739 doi "https://doi.org/10.1016/j.bmcl.2008.05.076" @default.
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