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- W2000507109 abstract "Le fentanyl est un analgésique opioïde de synthèse, lipophile, de courte durée d’action. Dans la douleur du cancer, il est couramment prescrit par voie transdermique pour traiter la douleur de fond. La forme injectable était jusqu’à présent réservée à l’anesthésie mais elle est désormais autorisée par voie intraveineuse ou sous-cutanée pour la prise en charge de douleurs réfractaires en cas d’échec ou d’intolérance à la morphine et à l’oxycodone. Des nouvelles formes galéniques transmuqueuses, buccales ou nasales ont fait preuve de leur efficacité dans la prise en charge des accès douloureux paroxystiques (ADP) ; la période de titration est souvent délicate car la dose requise pour un soulagement suffisant ne peut pas s’extrapoler à partir de la dose de fond. Cet article passe en revue les aspects pharmacocinétiques, pharmacodynamiques et l’efficacité clinique des ces différents modes d’administration. Fentanyl is a synthetic opioid analgesic with lipophilic, short-acting properties. In cancer-related pain, transdermic fentanyl is widely used for baseline pain. Injectable form was reserved to anaesthesia but is now available by intravenous or subcutaneous route in cases of refractory pain with failure or unmanageable adverse events after morphine or oxycodone. Buccal or intranasal transmucosal forms have shown efficacy for the management of breakthrough pain; titration period is necessary to determine the dose that produced satisfactory pain relief, which is not related to the baseline dose. This article reviews the pharmacokinetics, pharmacodynamics and clinical efficacy of these various forms of fentanyl." @default.
- W2000507109 created "2016-06-24" @default.
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- W2000507109 date "2011-12-01" @default.
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- W2000507109 title "Le fentanyl en soins palliatifs : de la pharmacologie à la clinique" @default.
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- W2000507109 doi "https://doi.org/10.1016/j.medpal.2010.11.005" @default.
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