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- W2001373281 endingPage "80" @default.
- W2001373281 startingPage "69" @default.
- W2001373281 abstract "Some neurones are endowed with receptors for endorphins and narcotic analgesics. Activation of these receptors results in a depression of the release of transmitter per impulse. It is currently believed that narcotic analgesics and endorphins depress the stimulus-induced influx of calcium (Ca2+) into the terminal and thereby modify the amount of the ion which triggers the release of the transmitter from intracellular stores. The influx of Ca2+ is largely governed by the Ca2+ channel, which opens during depolarization of the neuronal membrane either after an action potential (electrical stimulus) or in the presence of high extracellular potassium (K+) or nicotinic stimulants (chemical stimulus). The evoked influx of Ca2+ can be affected by a direct action on the Ca2+ channel or by primary actions on other membrane properties that subsequently regulate the Ca2+ channel. In many tissues narcotic analgesics and endorphins fail to inhibit transmitter release. This may be accounted for by the possibility that either such neurones lack presynaptic opiate receptors or that the function of existing receptors remains latent under the experimental conditions employed. Currently, there is insufficient evidence for endorphins physiologically modulating transmitter release." @default.
- W2001373281 created "2016-06-24" @default.
- W2001373281 creator A5013409891 @default.
- W2001373281 creator A5082722018 @default.
- W2001373281 date "1980-01-01" @default.
- W2001373281 modified "2023-10-14" @default.
- W2001373281 title "Candidate mechanisms for inhibition of neurotransmitter release by narcotic analgesics and endorphins" @default.
- W2001373281 cites W1488521817 @default.
- W2001373281 cites W1966611843 @default.
- W2001373281 cites W1968422198 @default.
- W2001373281 cites W1968464019 @default.
- W2001373281 cites W1969874446 @default.
- W2001373281 cites W1983628699 @default.
- W2001373281 cites W1983666386 @default.
- W2001373281 cites W1984912795 @default.
- W2001373281 cites W1985167215 @default.
- W2001373281 cites W1985763200 @default.
- W2001373281 cites W1985812179 @default.
- W2001373281 cites W1987558612 @default.
- W2001373281 cites W1992381290 @default.
- W2001373281 cites W1993652044 @default.
- W2001373281 cites W1994162219 @default.
- W2001373281 cites W1994535748 @default.
- W2001373281 cites W1994790318 @default.
- W2001373281 cites W1995437073 @default.
- W2001373281 cites W1995528444 @default.
- W2001373281 cites W1997396608 @default.
- W2001373281 cites W1999197169 @default.
- W2001373281 cites W1999825679 @default.
- W2001373281 cites W2003616417 @default.
- W2001373281 cites W2004681981 @default.
- W2001373281 cites W2005335314 @default.
- W2001373281 cites W2010051841 @default.
- W2001373281 cites W2011450946 @default.
- W2001373281 cites W2014358132 @default.
- W2001373281 cites W2014408481 @default.
- W2001373281 cites W2016726667 @default.
- W2001373281 cites W2021046666 @default.
- W2001373281 cites W2021847275 @default.
- W2001373281 cites W2022953311 @default.
- W2001373281 cites W2024933435 @default.
- W2001373281 cites W2026295851 @default.
- W2001373281 cites W2028160892 @default.
- W2001373281 cites W2031157126 @default.
- W2001373281 cites W2032024200 @default.
- W2001373281 cites W2032157777 @default.
- W2001373281 cites W2032352697 @default.
- W2001373281 cites W2032761582 @default.
- W2001373281 cites W2036580816 @default.
- W2001373281 cites W2038986594 @default.
- W2001373281 cites W2039462587 @default.
- W2001373281 cites W2040477003 @default.
- W2001373281 cites W2040494904 @default.
- W2001373281 cites W2040731339 @default.
- W2001373281 cites W2042781417 @default.
- W2001373281 cites W2050158678 @default.
- W2001373281 cites W2053243081 @default.
- W2001373281 cites W2057174730 @default.
- W2001373281 cites W2058611461 @default.
- W2001373281 cites W2061118062 @default.
- W2001373281 cites W2063605680 @default.
- W2001373281 cites W2067817117 @default.
- W2001373281 cites W2069498450 @default.
- W2001373281 cites W2069715753 @default.
- W2001373281 cites W2070275074 @default.
- W2001373281 cites W2070595451 @default.
- W2001373281 cites W2074303842 @default.
- W2001373281 cites W2075811628 @default.
- W2001373281 cites W2077361980 @default.
- W2001373281 cites W2080165573 @default.
- W2001373281 cites W2080753551 @default.
- W2001373281 cites W2081093344 @default.
- W2001373281 cites W2081807850 @default.
- W2001373281 cites W2084442692 @default.
- W2001373281 cites W2085642592 @default.
- W2001373281 cites W2086059365 @default.
- W2001373281 cites W2087273355 @default.
- W2001373281 cites W2088047884 @default.
- W2001373281 cites W2089033701 @default.
- W2001373281 cites W2089091308 @default.
- W2001373281 cites W2091044472 @default.
- W2001373281 cites W2094193448 @default.
- W2001373281 cites W2098656317 @default.
- W2001373281 cites W2140592883 @default.
- W2001373281 cites W2159852654 @default.
- W2001373281 cites W2165776873 @default.
- W2001373281 cites W2167846884 @default.
- W2001373281 cites W2179384912 @default.
- W2001373281 cites W2315341702 @default.
- W2001373281 cites W2420773174 @default.
- W2001373281 cites W2473976637 @default.
- W2001373281 cites W2580428309 @default.
- W2001373281 cites W4230454714 @default.
- W2001373281 cites W4233742517 @default.
- W2001373281 cites W4249225370 @default.
- W2001373281 cites W4254848357 @default.
- W2001373281 cites W4300495283 @default.
- W2001373281 cites W4318600690 @default.