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- W2003222044 abstract "In this study, the antipruritic effect of the methanol extract of Ganoderma lucidum (MEGL) was studied in mice. Oral administration of MEGL (10—1000 mg/kg) produced a dose-dependent inhibition of scratching, an itch-related response, induced by intradermal 5-hydroxytryptamine (5-HT) (100 nmol/site), α-methyl-5-HT (100 nmol/site), and proteinase-activated receptor-2 (PAR2)-activating peptide SLIGRL-NH2 (50 nmol/site). However, MEGL (100—1000 mg/kg) did not inhibit the scratching induced by histamine (100 nmol/site), substance P (100 nmol/site), and compound 48/80 (10 μg/site). These results raise the possibility that MEGL is effective against pruritus mediated by proteinases and 5-HT and that primary afferents expressing PAR2 and 5-HT2A receptors are the sites of its action." @default.
- W2003222044 created "2016-06-24" @default.
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- W2003222044 date "2010-01-01" @default.
- W2003222044 modified "2023-09-23" @default.
- W2003222044 title "Inhibitory Effect of Methanol Extract of Ganoderma lucidum on Acute Itch-Associated Responses in Mice" @default.
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- W2003222044 doi "https://doi.org/10.1248/bpb.33.909" @default.
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