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- W2003296498 abstract "Twenty-two compounds of substituted benzoylguanidine derivatives were designed and synthesized as potent NHE1 inhibitors. Twelve compounds showed more potent NHE1 inhibitory activity than cariporide. The activities of compounds 7e, 7h and 7j (IC50 = 0.073 ± 0.021, 0.084 ± 0.012 and 0.068 ± 0.021 nmol/L, respectively) were two orders of magnitude higher than that of cariporide (30.7 ± 2.5 nmol/L). Myocardial cells in vitro screening showed 7j had highlighted protective effect on cardiomyocytes subjected to hypoxia/reoxygenation. Thus it is valuable for further investigation." @default.
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- W2003296498 date "2010-06-01" @default.
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- W2003296498 title "MS144 MMP-10 UP-REGULATION IN PATIENTS WITH ENHANCED THROMBIN GENERATION: EVIDENCE IN VIVO AND IN VITRO OF A THROMBIN/CD40L MEDIATED MECHANISM" @default.
- W2003296498 doi "https://doi.org/10.1016/s1567-5688(10)70645-0" @default.
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