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- W2004366992 abstract "This study was carried out to determine both the effect of systemic paracetamol on the C-fibre evoked reflex activity, a test sensitive to centrally acting analgesic drugs, and the influence of an intrathecally administered 5HT3 receptor antagonist, tropisetron. Paracetamol (200, 300, 400 mg kg-1, i.v.) dose-dependently decreased (maximal effects -60 +/- 8%) the C-evoked responses for a duration of 90 min (for the lowest dose). This effect was totally suppressed by tropisetron (1 microgram, i.t.). These data confirm previous studies suggesting a central effect of this drug and demonstrate the involvement of a spinal 5HT3 mediated serotonergic mechanism." @default.
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- W2004366992 date "1995-07-01" @default.
- W2004366992 modified "2023-10-18" @default.
- W2004366992 title "Evidence of a central antinociceptive effect of paracetamol involving spinal 5HT3 receptors" @default.
- W2004366992 doi "https://doi.org/10.1097/00001756-199507310-00020" @default.
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