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- W2005281435 abstract "Abstract Molecular connectivity has been applied to the search of new compounds with activity against the protozoan Toxoplasma gondii, using a stepwise linear discriminant analysis (SLDA) which is able to classify a compound according its activity either as active or as inactive. Among the selected compounds, andrographolide and dibenzotiophene sulfone stand out, both with IC50 values lower than 1 μg/m1, which are comparable to these of drugs such as sulfamethoxazole, pyrimethamine and trimethoprim, with IC50 values equal to 1.1, 0.04 and 2.31 μg/ml, respectively. These results confirm the usefulness of our topological approach for the selection and design of new-lead drugs active against Toxoplasma gondii." @default.
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- W2005281435 title "Molecular Search of New Active Drugs Against<i>Toxoplasma Gondii</i>" @default.
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- W2005281435 doi "https://doi.org/10.1080/10629369908039165" @default.
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