Matches in SemOpenAlex for { <https://semopenalex.org/work/W2006746802> ?p ?o ?g. }
- W2006746802 endingPage "1145" @default.
- W2006746802 startingPage "1123" @default.
- W2006746802 abstract "17beta-Hydroxysteroid dehydrogenases (17beta-HSDs) mainly catalyze the reduction of C17-ketosteroids to their corresponding hydroxylated forms as well as the reverse reaction (oxidation). Able to convert inactive or less active steroid hormones into more potent ones and vice versa, certain 17beta-HSDs play a key role, especially in the regulation of estrogen and androgen levels. The therapeutic potential of this enzyme family, especially for the treatment of breast cancer, prostate cancer, acne and osteoporosis, then stimulated the development of inhibitors of 17beta-HSDs and important progress was achieved over the last years.This review article reports all patent applications related to the inhibitors of 17beta-HSDs, including some articles needed to complement the information presented.Readers will be informed about the role and function of 17beta-HSDs in the first section and about the history of inhibitor development in the second section. Furthermore, in the third and main section, the readers will learn about the structures of patented inhibitors originating from different companies and academic groups.The increase in the number of 17beta-HSD inhibitors reported in the last years augurs well for the future. The challenge is now to translate these results into clinical studies to allow determination of the therapeutic usefulness of 17beta-HSD inhibitors." @default.
- W2006746802 created "2016-06-24" @default.
- W2006746802 creator A5034301403 @default.
- W2006746802 date "2010-07-20" @default.
- W2006746802 modified "2023-09-30" @default.
- W2006746802 title "17β-Hydroxysteroid dehydrogenase inhibitors: a patent review" @default.
- W2006746802 cites W1503565230 @default.
- W2006746802 cites W1521693006 @default.
- W2006746802 cites W1543995018 @default.
- W2006746802 cites W1583940786 @default.
- W2006746802 cites W1601614768 @default.
- W2006746802 cites W1833278024 @default.
- W2006746802 cites W1926005362 @default.
- W2006746802 cites W1968886314 @default.
- W2006746802 cites W1970181773 @default.
- W2006746802 cites W1970687343 @default.
- W2006746802 cites W1971097859 @default.
- W2006746802 cites W1971318128 @default.
- W2006746802 cites W1977144806 @default.
- W2006746802 cites W1978187957 @default.
- W2006746802 cites W1978379711 @default.
- W2006746802 cites W1978895959 @default.
- W2006746802 cites W1980738399 @default.
- W2006746802 cites W1986420914 @default.
- W2006746802 cites W1988284423 @default.
- W2006746802 cites W1990047563 @default.
- W2006746802 cites W1990133984 @default.
- W2006746802 cites W1991430905 @default.
- W2006746802 cites W1994324783 @default.
- W2006746802 cites W1998102180 @default.
- W2006746802 cites W2001498773 @default.
- W2006746802 cites W2002837307 @default.
- W2006746802 cites W2007245161 @default.
- W2006746802 cites W2016183786 @default.
- W2006746802 cites W2016592632 @default.
- W2006746802 cites W2020259519 @default.
- W2006746802 cites W2020434370 @default.
- W2006746802 cites W2020881856 @default.
- W2006746802 cites W2024268846 @default.
- W2006746802 cites W2025397617 @default.
- W2006746802 cites W2026116352 @default.
- W2006746802 cites W2028085462 @default.
- W2006746802 cites W2028916314 @default.
- W2006746802 cites W2029030703 @default.
- W2006746802 cites W2031820370 @default.
- W2006746802 cites W2033568028 @default.
- W2006746802 cites W2043171291 @default.
- W2006746802 cites W2043188271 @default.
- W2006746802 cites W2043428993 @default.
- W2006746802 cites W2043974866 @default.
- W2006746802 cites W2046115334 @default.
- W2006746802 cites W2046238028 @default.
- W2006746802 cites W2048714965 @default.
- W2006746802 cites W2053405000 @default.
- W2006746802 cites W2055015510 @default.
- W2006746802 cites W2058878968 @default.
- W2006746802 cites W2061066255 @default.
- W2006746802 cites W2061646871 @default.
- W2006746802 cites W2062790615 @default.
- W2006746802 cites W2072243132 @default.
- W2006746802 cites W2072436322 @default.
- W2006746802 cites W2076068021 @default.
- W2006746802 cites W2077134485 @default.
- W2006746802 cites W2081285496 @default.
- W2006746802 cites W2081922333 @default.
- W2006746802 cites W2083318977 @default.
- W2006746802 cites W2087279497 @default.
- W2006746802 cites W2089418739 @default.
- W2006746802 cites W2094624406 @default.
- W2006746802 cites W2097678737 @default.
- W2006746802 cites W2107758429 @default.
- W2006746802 cites W2113409906 @default.
- W2006746802 cites W2116051622 @default.
- W2006746802 cites W2116838171 @default.
- W2006746802 cites W2117965089 @default.
- W2006746802 cites W2126846194 @default.
- W2006746802 cites W2127529986 @default.
- W2006746802 cites W2131642993 @default.
- W2006746802 cites W2145735545 @default.
- W2006746802 cites W2145801998 @default.
- W2006746802 cites W2148979187 @default.
- W2006746802 cites W2150653028 @default.
- W2006746802 cites W2152997446 @default.
- W2006746802 cites W2163801743 @default.
- W2006746802 cites W2168990617 @default.
- W2006746802 cites W2173684587 @default.
- W2006746802 cites W2261726786 @default.
- W2006746802 cites W2400271924 @default.
- W2006746802 cites W2412673684 @default.
- W2006746802 cites W2415785512 @default.
- W2006746802 cites W2426333224 @default.
- W2006746802 cites W2949747570 @default.
- W2006746802 cites W2952757175 @default.
- W2006746802 cites W3025410850 @default.
- W2006746802 cites W4211225750 @default.
- W2006746802 cites W4246234200 @default.
- W2006746802 cites W615323360 @default.
- W2006746802 cites W4211121400 @default.