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- W2007820163 startingPage "327" @default.
- W2007820163 abstract "Adenosine is an endogenous purine nucleoside that is an important metabolic sensing molecule. It is released during conditions of low oxygen delivery to tissues and organs to activate a range of effects in vascular tissues. Adenosine has a role in the vasculature by mediating vasodilation, vessel remodelling, cell proliferation as well as antiplatelet and inflammatory responses. Also, adenosine stimulates vasculogenesis and angiogenesis during wound healing and tumour growth. Currently, the clinical uses of adenosine are limited to treatment of supraventricular tachycardia or as a coronary vasodilator during radionuclide myocardial perfusion imaging. Due to the involvement of adenosine in various pathological conditions, the targeting of specific adenosine receptor (ADOR) subtypes in the vasculature using selective ADOR agonists or antagonists could have potential therapeutic benefit. However, the distribution of the receptors differs between species. Therefore, cross-species testing is essential to validate drug function. Keywords: Adenosine, adenosine receptors, adenosine metabolism, blood vessels, vasodilation, vessel remodelling." @default.
- W2007820163 created "2016-06-24" @default.
- W2007820163 creator A5012110713 @default.
- W2007820163 creator A5057765718 @default.
- W2007820163 date "2013-05-01" @default.
- W2007820163 modified "2023-10-17" @default.
- W2007820163 title "Vascular Adenosine Receptors; Potential Clinical Applications" @default.
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