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- W2007825231 abstract "The fact that SCH 23390, a selective dopamine (DA) D1 antagonist, blocks the effects of D2 agonists suggests a functional coupling of D1 and D2 receptors. Therefore, the binding of SCH 23390 to D2 receptors was investigated in vivo using 3H-N-n-propylnorapomorphine (NPA), a D2 agonist, and 3H-spiperone and 3H-raclopride, both D2 antagonists. SCH 23390 failed to inhibit 3H-spiperone or 3H-raclopride binding; however, SCH 23390 was relatively potent in inhibiting 3H-NPA binding. These results suggest that (some) antidopaminergic effects of SCH 23390 may result from antagonism of a D2 agonist conformation of the D2 receptor." @default.
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- W2007825231 date "2009-03-13" @default.
- W2007825231 modified "2023-09-27" @default.
- W2007825231 title "The Benzazepine, SCH 23390, Inhibits 3H-NPA Binding in Mouse Brain In Vivo" @default.
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- W2007825231 doi "https://doi.org/10.1111/j.1600-0773.1986.tb00175.x" @default.
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