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- W2009277746 abstract "The new conjugate, 177Lu-DOTA-8-Aoc-BBN[7–14]NH2, was prepared in high yield (≥95%) upon addition of 177LuCl3 to an aqueous solution (Ammonium Acetate) of DOTA-8-Aoc-BBN[7–14]NH2. The 177Lu-DOTA-8-Aoc-BBN[7–14]NH2-conjugate is stable over a wide range of pHs and does not undergo in vitro decomposition for ≤24h. Biodistribution studies of the 177Luconjugate were determined in tumor bearing (PC-3), SCID mice. Tumor uptake and retention values of 4.22 ± 1.09%ID/g, 3.03 ± 0.91%ID/g, and 1.54 ± 1.14%ID/g were obtained at 1, 4, and 24h, respectively." @default.
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- W2009277746 date "2001-05-01" @default.
- W2009277746 modified "2023-09-25" @default.
- W2009277746 title "Radiochemical investigations of 177Lu-DOTA-8-Aoc-BBN[7-14]NH2: A new gastrin releasing peptide receptor (GRPr) targeting radiopharma ceutical" @default.
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- W2009277746 doi "https://doi.org/10.1002/jlcr.25804401249" @default.
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