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- W2011056781 abstract "Efforts to improve the potency and physical properties of the aminopyridiopyrazinone class of PDE5 inhibitors through modification of the core ring system are described. Five new ring systems are evaluated and features that impart improved potency and improved solubility are delineated." @default.
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- W2011056781 date "2009-08-01" @default.
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- W2011056781 title "Investigation of aminopyridiopyrazinones as PDE5 inhibitors: Evaluation of modifications to the central ring system" @default.
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- W2011056781 doi "https://doi.org/10.1016/j.bmcl.2009.06.004" @default.
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