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- W2011736771 abstract "The success of early drug-discovery programs depends on the adequate combination of complementary and orthogonal technologies allowing hit/lead compounds to be optimized and improve therapeutic activity. Among the available biophysical methods, native MS recently emerged as an efficient method for compound-binding screening. Native MS is a highly sensitive and accurate screening technique. This review provides a description of the general approach and an overview of the possible characterization of ligand-binding properties. How native MS supports structure- and fragment-based drug research will also be discussed, with examples from the literature and internal developments. Native MS shows strong potential for in-depth characterization of ligand-binding properties. It is also a reliable screening technique in drug-discovery processes." @default.
- W2011736771 created "2016-06-24" @default.
- W2011736771 creator A5023284045 @default.
- W2011736771 creator A5041974331 @default.
- W2011736771 creator A5053461134 @default.
- W2011736771 creator A5060217867 @default.
- W2011736771 creator A5073068916 @default.
- W2011736771 date "2010-01-01" @default.
- W2011736771 modified "2023-09-26" @default.
- W2011736771 title "Native MS: an ’ESI‚ way to support structure- and fragment-based drug discovery" @default.
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