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- W2012095265 abstract "Interaction of sigma receptors with intracellular Ca2+ channel blocker and modulators was examined. Ryanodine and inositol 1,4,5-trisphosphate (IP3) did not inhibit [3H](+)-N-allylnormetazocine ([3H](+)-SKF-10047) binding to sigma receptors from either brain microsomal fractions or liver membrane extracts of the rat. However, the IP3 receptor antagonist heparin inhibited [3H](+)-SKF-10047 to sigma receptors in an uncompetitive manner with a Ki of 93 microM. These results suggest that sigma receptors may bear some relationship with IP3 receptor associated proteins or channels." @default.
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- W2012095265 title "IP3 receptor antagonist heparin uncompetitively inhibits [3H](+)-SKF-10047 binding to σ receptors" @default.
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- W2012095265 doi "https://doi.org/10.1016/0014-2999(96)00533-x" @default.
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