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- W2012503063 abstract "The discovery of GS-9451 is reported. Modification of the P3 cap and P2 quinoline with a series of solubilizing groups led to the identification of potent HCV NS3 protease inhibitors with greatly improved pharmacokinetic properties in rats, dogs and monkeys." @default.
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- W2012503063 date "2012-04-01" @default.
- W2012503063 modified "2023-10-11" @default.
- W2012503063 title "Discovery of GS-9451: An acid inhibitor of the hepatitis C virus NS3/4A protease" @default.
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- W2012503063 doi "https://doi.org/10.1016/j.bmcl.2012.01.017" @default.
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