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- W2012966353 endingPage "414" @default.
- W2012966353 startingPage "405" @default.
- W2012966353 abstract "Delta opioid receptors represent a promising target for the development of novel analgesics. A number of tools have been developed recently that have significantly improved our knowledge of δ receptor function in pain control. These include several novel δ agonists with potent analgesic properties, and genetic mouse models with targeted mutations in the δ opioid receptor gene. Also, recent findings have further documented the regulation of δ receptor function at cellular level, which impacts on the pain-reducing activity of the receptor. These regulatory mechanisms occur at transcriptional and post-translational levels, along agonist-induced receptor activation, signaling and trafficking, or in interaction with other receptors and neuromodulatory systems. All these tools for in-vivo research, and proposed mechanisms at molecular level, have tremendously increased our understanding of δ receptor physiology, and contribute to designing innovative strategies for the treatment of chronic pain and other diseases such as mood disorders." @default.
- W2012966353 created "2016-06-24" @default.
- W2012966353 creator A5031112700 @default.
- W2012966353 creator A5041985407 @default.
- W2012966353 date "2011-09-01" @default.
- W2012966353 modified "2023-10-08" @default.
- W2012966353 title "Delta opioid receptor analgesia" @default.
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