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- W2013362029 abstract "SAR exploration at C-6 and C-8 positions of the tricyclic sulfone series was carried out. Several functional groups were found to be well tolerated at C-6 and C-8 positions. Selective combination of C-6 and C-8 modification resulted in new tricyclic sulfone analogs with efficacy in in vivo mouse Aβ(40) lowering model." @default.
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- W2013362029 date "2011-06-01" @default.
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- W2013362029 title "Synthesis and SAR study of tricyclic sulfones as γ-secretase inhibitors: C-6 and C-8 positions" @default.
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- W2013362029 doi "https://doi.org/10.1016/j.bmcl.2011.03.094" @default.
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