Matches in SemOpenAlex for { <https://semopenalex.org/work/W2013434401> ?p ?o ?g. }
- W2013434401 endingPage "77" @default.
- W2013434401 startingPage "66" @default.
- W2013434401 abstract "Parasitic diseases cause significant global morbidity and mortality, particularly in underdeveloped regions of the world. Malaria alone causes ∼800 000 deaths each year, with children and pregnant women being at highest risk. There is no licensed vaccine available for any human parasitic disease and drug resistance is compromising the efficacy of many available anti-parasitic drugs. This is driving drug discovery research on new agents with novel modes of action. Histone deacetylase (HDAC) inhibitors are being investigated as drugs for a range of diseases, including cancers and infectious diseases such as HIV/AIDS, and several parasitic diseases. This review focuses on the current state of knowledge of HDAC inhibitors targeted to the major human parasitic diseases malaria, schistosomiasis, trypanosomiasis, toxoplasmosis and leishmaniasis. Insights are provided into the unique challenges that will need to be considered if HDAC inhibitors are to be progressed towards clinical development as potential new anti-parasitic drugs." @default.
- W2013434401 created "2016-06-24" @default.
- W2013434401 creator A5039640617 @default.
- W2013434401 creator A5053330477 @default.
- W2013434401 creator A5084779683 @default.
- W2013434401 date "2011-11-29" @default.
- W2013434401 modified "2023-10-03" @default.
- W2013434401 title "HDAC inhibitors in parasitic diseases" @default.
- W2013434401 cites W1513489828 @default.
- W2013434401 cites W1587810042 @default.
- W2013434401 cites W1963724149 @default.
- W2013434401 cites W1963775811 @default.
- W2013434401 cites W1964317228 @default.
- W2013434401 cites W1966000993 @default.
- W2013434401 cites W1969180448 @default.
- W2013434401 cites W1972533251 @default.
- W2013434401 cites W1977082621 @default.
- W2013434401 cites W1978455510 @default.
- W2013434401 cites W1980654946 @default.
- W2013434401 cites W1983970357 @default.
- W2013434401 cites W1988473164 @default.
- W2013434401 cites W1988688335 @default.
- W2013434401 cites W1990395956 @default.
- W2013434401 cites W1990801507 @default.
- W2013434401 cites W1991094038 @default.
- W2013434401 cites W1992581726 @default.
- W2013434401 cites W1993176720 @default.
- W2013434401 cites W1997959217 @default.
- W2013434401 cites W1999536542 @default.
- W2013434401 cites W2001101815 @default.
- W2013434401 cites W2004894632 @default.
- W2013434401 cites W2006461939 @default.
- W2013434401 cites W2007772408 @default.
- W2013434401 cites W2008953417 @default.
- W2013434401 cites W2009715792 @default.
- W2013434401 cites W2009717402 @default.
- W2013434401 cites W2011326960 @default.
- W2013434401 cites W2013588595 @default.
- W2013434401 cites W2013644391 @default.
- W2013434401 cites W2014275882 @default.
- W2013434401 cites W2021926390 @default.
- W2013434401 cites W2023411386 @default.
- W2013434401 cites W2024425375 @default.
- W2013434401 cites W2024639033 @default.
- W2013434401 cites W2024804690 @default.
- W2013434401 cites W2027452158 @default.
- W2013434401 cites W2029763251 @default.
- W2013434401 cites W2030064289 @default.
- W2013434401 cites W2036605603 @default.
- W2013434401 cites W2037168603 @default.
- W2013434401 cites W2041036553 @default.
- W2013434401 cites W2043634732 @default.
- W2013434401 cites W2046105178 @default.
- W2013434401 cites W2046144222 @default.
- W2013434401 cites W2048289333 @default.
- W2013434401 cites W2049453822 @default.
- W2013434401 cites W2051933643 @default.
- W2013434401 cites W2052703240 @default.
- W2013434401 cites W2059301290 @default.
- W2013434401 cites W2062950876 @default.
- W2013434401 cites W2064138320 @default.
- W2013434401 cites W2066544271 @default.
- W2013434401 cites W2066887945 @default.
- W2013434401 cites W2066910902 @default.
- W2013434401 cites W2067888376 @default.
- W2013434401 cites W2070433411 @default.
- W2013434401 cites W2077747170 @default.
- W2013434401 cites W2082857661 @default.
- W2013434401 cites W2082946800 @default.
- W2013434401 cites W2083280521 @default.
- W2013434401 cites W2089848238 @default.
- W2013434401 cites W2094169801 @default.
- W2013434401 cites W2101092227 @default.
- W2013434401 cites W2102155970 @default.
- W2013434401 cites W2103665811 @default.
- W2013434401 cites W2104945888 @default.
- W2013434401 cites W2105688902 @default.
- W2013434401 cites W2112047656 @default.
- W2013434401 cites W2114987890 @default.
- W2013434401 cites W2124258829 @default.
- W2013434401 cites W2131163323 @default.
- W2013434401 cites W2131249903 @default.
- W2013434401 cites W2132006467 @default.
- W2013434401 cites W2138699994 @default.
- W2013434401 cites W2146180663 @default.
- W2013434401 cites W2149232833 @default.
- W2013434401 cites W2151243604 @default.
- W2013434401 cites W2152295227 @default.
- W2013434401 cites W2156022009 @default.
- W2013434401 cites W2156995961 @default.
- W2013434401 cites W2158178080 @default.
- W2013434401 cites W2159278252 @default.
- W2013434401 cites W2161311583 @default.
- W2013434401 cites W2162414508 @default.
- W2013434401 cites W2163062563 @default.
- W2013434401 cites W2164365774 @default.
- W2013434401 cites W2164689318 @default.
- W2013434401 cites W2166299057 @default.