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- W2015535421 abstract "Anti-HIV peptides with inhibitory activity against HIV-1 integrase (IN) have been found in overlapping peptide libraries derived from HIV-1 gene products. In a strand transfer assay using IN, inhibitory active peptides with certain sequential motifs related to Vpr- and Env-derived peptides were found. The addition of an octa-arginyl group to the inhibitory peptides caused a remarkable inhibition of the strand transfer and 3′-end-processing reactions catalyzed by IN and significant inhibition against HIV replication." @default.
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- W2015535421 date "2010-06-29" @default.
- W2015535421 modified "2023-10-16" @default.
- W2015535421 title "Peptide HIV-1 Integrase Inhibitors from HIV-1 Gene Products" @default.
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- W2015535421 doi "https://doi.org/10.1021/jm1003528" @default.
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