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- W2015996312 abstract "A series of alkyne-containing type II inhibitors with potent inhibitory activity of T315I Bcr-Abl has been identified. The most active compound 4 exhibits an EC(50) of less than 1 nM against wild-type Bcr-Abl and an EC(50) of 10 nM against T315I mutant but is broadly active against a number of other kinases." @default.
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- W2015996312 title "Broad spectrum alkynyl inhibitors of T315I Bcr-Abl" @default.
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- W2015996312 doi "https://doi.org/10.1016/j.bmcl.2010.05.043" @default.
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