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- W2016079923 abstract "Evidence exists to implicate the monoamine histamine in the control of arousal and cognitive functions. Antagonists of H3 receptors are postsynaptic and presynaptic modulators of neural transmission in a variety of neuronal circuits relevant to cognition. Accumulating neuroanatomical, neurochemical, pharmacological, and behavioral data support the idea that H3 receptor antagonists may function to improve cognitive performances in disease states (e.g., Alzheimer's disease and mild cognitive impairment states). Thus, H3 receptor antagonists have been shown to increase performance in attention and memory tests in nonhuman experiments and prevent the degradation in performances produced by scopolamine, MK-801, or age. In contrast, agonists of the H3 receptor generally produce cognitive impairing effects in animal models. The role of H3 receptors in these behavioral effects is substantiated by data indicating a central origin for their effects, the selectivity of some of the H3 receptor antagonists studied, and the pharmacological modification of effects of H3 receptor antagonists by selective H3 receptor agonists. Data and issues that challenge the potential role for H3 receptor antagonists in cognitive processes are also critically reviewed. H3 receptor antagonists may also have therapeutic value in the management of obesity, pain, sleep disorders, schizophrenia, and attention deficit hyperactivity disorder." @default.
- W2016079923 created "2016-06-24" @default.
- W2016079923 creator A5022661281 @default.
- W2016079923 creator A5090899159 @default.
- W2016079923 date "2004-07-01" @default.
- W2016079923 modified "2023-10-18" @default.
- W2016079923 title "Selective histamine H3 receptor antagonists for treatment of cognitive deficiencies and other disorders of the central nervous system" @default.
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