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- W2016216356 abstract "CYP2C enzymes are responsible for the oxidative metabolism of a diverse number of drugs for the treatment of type 2 diabetes mellitus, a severe metabolic disorder with high prevalence. Various clinical studies found the close association between CYP2C polymorphisms and altered pharmacokinetics, toxicological profiles, and drug-drug interactions of antidiabetic drugs. In this brief review, we discussed the impact of CYP2C polymorphisms on the metabolic fate of small-molecule antidiabetics including sulfonylureas, meglitinides, thiazolidinediones, gliptins, and gliflozins, with the key drug-protein molecular interactions highlighted." @default.
- W2016216356 created "2016-06-24" @default.
- W2016216356 creator A5071208746 @default.
- W2016216356 creator A5081011722 @default.
- W2016216356 date "2011-11-01" @default.
- W2016216356 modified "2023-10-01" @default.
- W2016216356 title "Impact of genetic polymorphisms of cytochrome P450 2 C (CYP2C) enzymes on the drug metabolism and design of antidiabetics" @default.
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- W2016216356 doi "https://doi.org/10.1016/j.cbi.2011.08.011" @default.
- W2016216356 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/21939641" @default.
- W2016216356 hasPublicationYear "2011" @default.
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