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- W2016340819 abstract "ExoU is a potent virulence factor of Pseudomonas aeruginosa and is considered a potential therapeutic target. In order to discover novel ExoU inhibitors, we screened an in-house chemical library utilizing a yeast-based screening system. Some sulfonamides displayed significant activity without nonspecific cytotoxicity. We describe a series of sulfonamides as novel ExoU inhibitors, along with a brief structure–activity relationship." @default.
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- W2016340819 date "2014-08-01" @default.
- W2016340819 modified "2023-10-01" @default.
- W2016340819 title "Identification of arylsulfonamides as ExoU inhibitors" @default.
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- W2016340819 doi "https://doi.org/10.1016/j.bmcl.2014.06.064" @default.
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