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- W2017026208 abstract "The beta-carbolines harmane and norharmane competitively inhibit [3H]flunitrazepam ([3H]FNZ) binding to deoxycholate-solubilized benzodiazepine receptors from calf cerebral cortex, with Ki in the micromolar range [3H]Propyl-beta-carboline-3-carboxylate ([3H]PrCC) binds to the soluble receptors with an affinity similar to its binding to particulate receptors (0.41 nM vs 0.48 nM, respectively). The component that binds [3H]PrCC displays a sedimentation profile on sucrose gradient centrifugation similar to that of [3H]FNZ binding component (sedimentation coefficient about 11S)." @default.
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- W2017026208 date "1981-11-01" @default.
- W2017026208 modified "2023-09-27" @default.
- W2017026208 title "β-Carboline binding to deoxycholate solubilized benzodiazepine receptors from calf cerebral cortex" @default.
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- W2017026208 doi "https://doi.org/10.1016/0304-3940(81)90153-1" @default.
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