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- W2017059175 abstract "A series of pyrimidinopyridones has been designed, synthesized and shown to be potent and selective inhibitors of the FMS tyrosine kinase. Introduction of an amide substituent at the 6-position of the pyridone core resulted in a significant potency increase. Compound 24 effectively inhibited in vivo LPS-induced TNF in mice greater than 80%." @default.
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- W2017059175 date "2008-04-01" @default.
- W2017059175 modified "2023-09-23" @default.
- W2017059175 title "Design and synthesis of a pyrido[2,3-d]pyrimidin-5-one class of anti-inflammatory FMS inhibitors" @default.
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- W2017059175 doi "https://doi.org/10.1016/j.bmcl.2008.02.070" @default.
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