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- W2019118611 abstract "A series of novel 5-aminomethyl-1H-benzimidazole based inhibitors of Itk were prepared. Structure-activity relationships, selectivity and cell activity are reported for this series. Compound 2, a potent and selective antagonist of Itk, inhibited anti-CD3 antibody induced IL-2 production in vivo in mice." @default.
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- W2019118611 date "2008-10-01" @default.
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- W2019118611 title "5-Aminomethyl-1H-benzimidazoles as orally active inhibitors of inducible T-cell kinase (Itk)" @default.
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- W2019118611 doi "https://doi.org/10.1016/j.bmcl.2008.09.016" @default.
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