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- W2019156684 abstract "The effects of botulinum C2 toxin, which ADP-ribosylates actin, were studied on the stimulated histamine release of rat peritoneal mast cells. Treatment of mast cells with botulinum C2 toxin for 4 h inhibited histamine release stimulated by compound 48/80 or MCD-peptide maximally by about 50%. A half-maximal and maximal inhibition occurred at about 30 and 450 ng/ml botulinum C2 toxin. At similar concentrations the toxin ADP-ribosylated actin in intact mast cells. Botulinum C2 toxin largely impaired the histamine release stimulated by 12-<i>O</i>-tetradecanoylphorbol-13-acetate but not by the ionophore A23187. The data indicate that botulinum C2 toxin partially inhibits the stimulated histamine release and suggest that actin is involved in the stimulus-secretion coupling in mast cells." @default.
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- W2019156684 date "1987-01-01" @default.
- W2019156684 modified "2023-09-23" @default.
- W2019156684 title "Inhibition of Histamine Release from Rat Mast Cells by Botulinum C2 Toxin" @default.
- W2019156684 doi "https://doi.org/10.1159/000234453" @default.
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