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- W2020147653 abstract "A possible interaction of the antihypertensive drug, urapidil with beta-adrenoceptors was investigated in a guinea-pig ventricular membrane preparation. Urapidil at concentrations above 1 microM antagonized the isoproterenol-induced stimulation of adenylate cyclase activity. Urapidil 10 microM shifted the concentration-response curve for isoproterenol in a parallel manner to the right by a factor of 16. Urapidil competed with specific beta-adrenoceptor binding of [125I]iodocyanopindolol with an IC50 of 12 microM. Since the affinity of urapidil to beta-adrenoceptors appeared rather low, any beta-adrenoceptor blocking property may be of relevance in vivo at high dosages only." @default.
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- W2020147653 date "1984-09-01" @default.
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- W2020147653 title "Interaction of the antihypertensive drug urapidil with cardiac β-adrenoceptors in vitro" @default.
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- W2020147653 doi "https://doi.org/10.1016/0014-2999(84)90385-6" @default.
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