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- W2020170393 abstract "Spirodiketopiperazine-based CCR5 antagonists, showing improved pharmacokinetic profiles without reduction in antagonist activity, were designed and synthesized. We also demonstrate the anti-HIV activity of a representative compound 12, as measured in a p24 assay." @default.
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- W2020170393 date "2010-01-01" @default.
- W2020170393 modified "2023-10-09" @default.
- W2020170393 title "Spirodiketopiperazine-based CCR5 antagonists: Improvement of their pharmacokinetic profiles" @default.
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- W2020170393 doi "https://doi.org/10.1016/j.bmcl.2009.11.018" @default.
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