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- W2022131049 abstract "Insecticidal bioassays on Plutella xylostella (Linneaus) of an oxadiazine insecticide indoxacarb and its N-decarbomethoxylated metabolite (DCJW), and their modulation of voltage-gated sodium channels in rat dorsal root ganglion neurons were examined. No significant difference was observed in insecticidal activity between indoxacarb and DCJW in ingestion and contact tests. In patch-clamp experiments, both indoxacarb and DCJW suppressed the peak sodium currents in a time- and dose-dependent manner. DCJW at 1 μM blocked the sodium currents to 62.7±3.0% (n=5) of the control after 25 min of bath application. In contrast, in the presence of 1 μM indoxacarb, currents were blocked to 4.5±0.6% (n=4) of control. Thus, the potency of DCJW in blocking sodium currents was higher than that of indoxacarb in rat dorsal root ganglion neurons." @default.
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- W2022131049 date "2001-01-01" @default.
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- W2022131049 title "Insecticidal activity of oxadiazine insecticide indoxacarb and its N-decarbomethoxylated metabolite and their modulations of voltage-gated sodium channels." @default.
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- W2022131049 doi "https://doi.org/10.1303/aez.2001.381" @default.
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