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- W2022149323 abstract "Novel thrombin inhibitors incorporating thienylamidine at the P1 position were designed and synthesized. These compounds are potent, trypsin-selective and efficacious in the rat model of venous thrombosis. The proposed P1 binding mode in the thrombin active site was confirmed by X-ray crystallographic analysis." @default.
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- W2022149323 title "Potent and efficacious thienylamidine-incorporated thrombin inhibitors" @default.
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