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- W2022284188 abstract "In exploring for templates to devise novel antagonists for the integrins α4β1 and α4β7, was a series of compounds identified possessing a 1,2,4-triazolo[2,3-a]pyrrole structural subunit. Compound 11, for example, was found to antagonize α4β1-VCAM-1 and α4β7-MAdCAM-1 adhesion with IC50 values of 80 and 20 nM, respectively. Keywords: Integrin receptors, VCAM-1, arylcarboxamido, pharmacokinetics, LDT-based peptides" @default.
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- W2022284188 date "2005-12-01" @default.
- W2022284188 modified "2023-09-23" @default.
- W2022284188 title "Synthesis and Biological Evaluation of 1,2,4-Triazolo[2,3-a]pyrrole Derivatives as Alpha-4 ( α4) Integrin Antagonists" @default.
- W2022284188 doi "https://doi.org/10.2174/157018005774717280" @default.
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