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- W2022392198 abstract "TAK-778, a novel synthetic 3-benzothiepin derivative, stimulates the formation of cartilaginous nodules in mouse chondroprogenitor-like ATDC5 cells in vitro in association with upregulation of the gene expression of transforming growth factor-beta(2), but not bone morphogenetic protein-4 and insulin-like growth factor-I. One-shot injection of the TAK-778-containing sustained-release microcapsules accelerated the repair process of the full thickness defects of articular cartilage in rabbit knees. Our in vitro and in vivo results indicate that TAK-778 may be a therapeutically useful synthetic agent for articular cartilage repair." @default.
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- W2022392198 date "1999-07-01" @default.
- W2022392198 modified "2023-09-24" @default.
- W2022392198 title "TAK-778, a Novel Synthetic 3-Benzothiepin Derivative, Promotes Chondrogenesis in Vitro and in Vivo" @default.
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- W2022392198 doi "https://doi.org/10.1006/bbrc.1999.0991" @default.
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