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- W2022603937 abstract "In silico screening in combination with activity-based protein profiling as a strategy for discovering selective hits in complex brain proteome is presented by M. van der Stelt et al. in their Communication on page 12081 ff. A common starting point was used for the generation of both the pharmacophore model and the activity-based probe. This resulted in the identification of a novel class of diacylglycerol lipase-α inhibitors with high selectivity in the brain proteome." @default.
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- W2022603937 date "2013-11-07" @default.
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- W2022603937 title "Inside Back Cover: Development of an Activity-Based Probe and In Silico Design Reveal Highly Selective Inhibitors for Diacylglycerol Lipase-α in Brain (Angew. Chem. Int. Ed. 46/2013)" @default.
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