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- W2022771372 abstract "Abstract: Interaction of Li + with the voltage‐dependent Na + channel has been analyzed in neuroblastoma × glioma hybrid cells. The cells were able to generate action potentials in media containing Li + instead of Na + . The uptake of Li + into the hybrid cells was investigated for the pharmacological analysis of Li + permeation through voltage‐dependent Na + channels. Veratridine and acionitine increased the uptake of Li + to the same degree (EC 50 30 μ M ). This increase was blocked by tetrodotoxin (IC 50 20 n M ). Veratridine and aconitine did not act synergistically; however, the veratridine‐stimulated influx was further enhanced by the toxin of the scorpion Leiurus quinquestriatus (EC 50 0.06 μg/ml). This stimulation was also blocked by tetrodotoxin. Thus, the voltage‐dependent Na + channel of the hybrid cells accepts both Li + and Na + in a similar manner." @default.
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- W2022771372 date "1982-07-01" @default.
- W2022771372 modified "2023-10-15" @default.
- W2022771372 title "Pharmacological and Electrophysiological Characterization of Lithium Ion Flux Through the Action Potential Sodium Channel in Neuroblastoma × Glioma Hybrid Cells" @default.
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- W2022771372 doi "https://doi.org/10.1111/j.1471-4159.1982.tb04723.x" @default.
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