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- W2022785868 abstract "The bradykinin B1 receptor is rapidly induced after inflammation or tissue trauma and appears to play an important role in the maintenance of hyperalgesia in inflammatory conditions. Here, we describe the optimization process to identify novel, potent non-peptide human B1 receptor antagonists based on a 2-alkylamino-5-sulfamoylbenzamide core. Optimized derivatives are selective, functional B1 antagonists with low nanomolar affinity and exhibit oral bioavailability in animals." @default.
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- W2022785868 date "2004-08-10" @default.
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- W2022785868 title "Potent and Orally Bioavailable Non-Peptide Antagonists at the Human Bradykinin B<sub>1</sub> Receptor Based on a 2-Alkylamino-5-sulfamoylbenzamide Core" @default.
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- W2022785868 doi "https://doi.org/10.1021/jm049747g" @default.
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