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- W2022896675 abstract "To date treatment of trypanosomiasis urgently requires new effective and non-toxic drugs. The article covers some of the achievements in the search for new antitrypanosomal agents; also the “validated” biological targets used in the antitrypanosomal agents design are outlined. The major part of the manuscript focuses on the synthetic small molecules, such as thiosemicarbazone and thiazole (as their cyclic analogues) derivatives, benzofuran derivatives, heterocycles bearing nitro group etc. Also, the attractiveness of metal complexes and well known drugs as sources for antitrypanosomal agent design is discussed." @default.
- W2022896675 created "2016-06-24" @default.
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- W2022896675 date "2014-10-01" @default.
- W2022896675 modified "2023-09-25" @default.
- W2022896675 title "Trends in research of antitrypanosomal agents among synthetic heterocycles" @default.
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- W2022896675 doi "https://doi.org/10.1016/j.ejmech.2014.07.092" @default.
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