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- W2023115772 endingPage "nrs.06010" @default.
- W2023115772 startingPage "nrs.06010" @default.
- W2023115772 abstract "Androgen receptor (AR) plays a critical role in the function of several organs including primary and accessory sexual organs, skeletal muscle, and bone, making it a desirable therapeutic target. Selective androgen receptor modulators (SARMs) bind to the AR and demonstrate osteo- and myo-anabolic activity; however, unlike testosterone and other anabolic steroids, these nonsteroidal agents produce less of a growth effect on prostate and other secondary sexual organs. SARMs provide therapeutic opportunities in a variety of diseases, including muscle wasting associated with burns, cancer, or end-stage renal disease, osteoporosis, frailty, and hypogonadism. This review summarizes the current standing of research and development of SARMs, crystallography of AR with SARMs, plausible mechanisms for their action and the potential therapeutic indications for this emerging class of drugs." @default.
- W2023115772 created "2016-06-24" @default.
- W2023115772 creator A5002243266 @default.
- W2023115772 creator A5016676195 @default.
- W2023115772 creator A5065375417 @default.
- W2023115772 creator A5067659573 @default.
- W2023115772 creator A5082023270 @default.
- W2023115772 date "2008-01-01" @default.
- W2023115772 modified "2023-10-16" @default.
- W2023115772 title "Selective androgen receptor modulators in preclinical and clinical development" @default.
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