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- W2023155850 abstract "A series of alkenyl indazoles were synthesized and evaluated in Aurora kinase enzyme assays. Several promising leads were optimized for selectivity towards Aurora B. Excellent binding affinity and good selectivity were achieved with optimized compounds in isolated Aurora subfamily assays." @default.
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- W2023155850 date "2010-04-01" @default.
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- W2023155850 title "Synthesis and evaluation of alkenyl indazoles as selective Aurora kinase inhibitors" @default.
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- W2023155850 doi "https://doi.org/10.1016/j.bmcl.2010.03.018" @default.
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