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- W2023361711 abstract "ABSTRACT The in vitro and in vivo activities of DW286, a novel fluoronaphthyridone with potent antibacterial activity, were compared with those of ciprofloxacin, gemifloxacin, sparfloxacin, and trovafloxacin. Against gram-positive bacteria, such as Staphylococcus aureus , Staphylococcus epidermidis , Streptococcus pneumoniae , and Enterococcus faecalis , the in vitro activity of DW286 was stronger than that of any other reference antibiotic. Against gram-negative bacteria, the activity of DW286 was similar to those of trovafloxacin and gemifloxacin but was weaker than that of ciprofloxacin. In a mouse systemic infection caused by three S. aureus strains, including methicillin-resistant S. aureus and quinolone-resistant S. aureus (QRSA), DW286 demonstrated the most potent activity, as found in vitro. Specially, DW286 is ≥8-fold more active against QRSA than the other fluoroquinolones. And the 50% protective doses for DW286 were correspondent with the in vitro activities." @default.
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- W2023361711 date "2002-09-01" @default.
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- W2023361711 title "In Vitro and In Vivo Antibacterial Activities of DW286, a New Fluoronaphthyridone Antibiotic" @default.
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- W2023361711 doi "https://doi.org/10.1128/aac.46.9.3071-3074.2002" @default.
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