Matches in SemOpenAlex for { <https://semopenalex.org/work/W2023454328> ?p ?o ?g. }
- W2023454328 endingPage "4295" @default.
- W2023454328 startingPage "4292" @default.
- W2023454328 abstract "This Letter discloses a series of 2-aminothiadiazole amides as selective EP(3) receptor antagonists. SAR optimization resulted in compounds with excellent functional activity in vitro. In addition, efforts to optimize DMPK properties in the rat are discussed. These efforts have resulted in the identification of potent, selective EP(3) receptor antagonists with excellent DMPK properties suitable for in vivo studies." @default.
- W2023454328 created "2016-06-24" @default.
- W2023454328 creator A5002551455 @default.
- W2023454328 creator A5007001805 @default.
- W2023454328 creator A5017578361 @default.
- W2023454328 creator A5020804233 @default.
- W2023454328 creator A5033973304 @default.
- W2023454328 creator A5034338625 @default.
- W2023454328 creator A5035411478 @default.
- W2023454328 creator A5037055416 @default.
- W2023454328 creator A5040067540 @default.
- W2023454328 creator A5058498730 @default.
- W2023454328 creator A5059655155 @default.
- W2023454328 creator A5078969103 @default.
- W2023454328 creator A5082703411 @default.
- W2023454328 creator A5091082571 @default.
- W2023454328 date "2009-08-01" @default.
- W2023454328 modified "2023-10-03" @default.
- W2023454328 title "Discovery of novel aminothiadiazole amides as selective EP3 receptor antagonists" @default.
- W2023454328 cites W1575388506 @default.
- W2023454328 cites W1647648618 @default.
- W2023454328 cites W1972643685 @default.
- W2023454328 cites W1974560730 @default.
- W2023454328 cites W1982309054 @default.
- W2023454328 cites W1993098410 @default.
- W2023454328 cites W1998798039 @default.
- W2023454328 cites W2009194925 @default.
- W2023454328 cites W2010977040 @default.
- W2023454328 cites W2029007266 @default.
- W2023454328 cites W2036754185 @default.
- W2023454328 cites W2038410983 @default.
- W2023454328 cites W2047770704 @default.
- W2023454328 cites W2071408538 @default.
- W2023454328 cites W2077603983 @default.
- W2023454328 cites W2080745027 @default.
- W2023454328 cites W2086145069 @default.
- W2023454328 cites W2121612337 @default.
- W2023454328 cites W2122172741 @default.
- W2023454328 cites W2122258650 @default.
- W2023454328 cites W2128173433 @default.
- W2023454328 cites W2129746956 @default.
- W2023454328 cites W2175319049 @default.
- W2023454328 cites W2333479422 @default.
- W2023454328 cites W4248634331 @default.
- W2023454328 doi "https://doi.org/10.1016/j.bmcl.2009.05.074" @default.
- W2023454328 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/19487124" @default.
- W2023454328 hasPublicationYear "2009" @default.
- W2023454328 type Work @default.
- W2023454328 sameAs 2023454328 @default.
- W2023454328 citedByCount "19" @default.
- W2023454328 countsByYear W20234543282012 @default.
- W2023454328 countsByYear W20234543282013 @default.
- W2023454328 countsByYear W20234543282014 @default.
- W2023454328 countsByYear W20234543282015 @default.
- W2023454328 countsByYear W20234543282016 @default.
- W2023454328 countsByYear W20234543282017 @default.
- W2023454328 countsByYear W20234543282018 @default.
- W2023454328 crossrefType "journal-article" @default.
- W2023454328 hasAuthorship W2023454328A5002551455 @default.
- W2023454328 hasAuthorship W2023454328A5007001805 @default.
- W2023454328 hasAuthorship W2023454328A5017578361 @default.
- W2023454328 hasAuthorship W2023454328A5020804233 @default.
- W2023454328 hasAuthorship W2023454328A5033973304 @default.
- W2023454328 hasAuthorship W2023454328A5034338625 @default.
- W2023454328 hasAuthorship W2023454328A5035411478 @default.
- W2023454328 hasAuthorship W2023454328A5037055416 @default.
- W2023454328 hasAuthorship W2023454328A5040067540 @default.
- W2023454328 hasAuthorship W2023454328A5058498730 @default.
- W2023454328 hasAuthorship W2023454328A5059655155 @default.
- W2023454328 hasAuthorship W2023454328A5078969103 @default.
- W2023454328 hasAuthorship W2023454328A5082703411 @default.
- W2023454328 hasAuthorship W2023454328A5091082571 @default.
- W2023454328 hasConcept C114373084 @default.
- W2023454328 hasConcept C150903083 @default.
- W2023454328 hasConcept C170493617 @default.
- W2023454328 hasConcept C185592680 @default.
- W2023454328 hasConcept C193042331 @default.
- W2023454328 hasConcept C202751555 @default.
- W2023454328 hasConcept C207001950 @default.
- W2023454328 hasConcept C21951064 @default.
- W2023454328 hasConcept C55493867 @default.
- W2023454328 hasConcept C86803240 @default.
- W2023454328 hasConcept C98274493 @default.
- W2023454328 hasConceptScore W2023454328C114373084 @default.
- W2023454328 hasConceptScore W2023454328C150903083 @default.
- W2023454328 hasConceptScore W2023454328C170493617 @default.
- W2023454328 hasConceptScore W2023454328C185592680 @default.
- W2023454328 hasConceptScore W2023454328C193042331 @default.
- W2023454328 hasConceptScore W2023454328C202751555 @default.
- W2023454328 hasConceptScore W2023454328C207001950 @default.
- W2023454328 hasConceptScore W2023454328C21951064 @default.
- W2023454328 hasConceptScore W2023454328C55493867 @default.
- W2023454328 hasConceptScore W2023454328C86803240 @default.
- W2023454328 hasConceptScore W2023454328C98274493 @default.
- W2023454328 hasIssue "15" @default.
- W2023454328 hasLocation W20234543281 @default.
- W2023454328 hasLocation W20234543282 @default.
- W2023454328 hasOpenAccess W2023454328 @default.