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- W2023786112 abstract "Nonmonotonic concentration response relationships are frequently observed for endocrine active ligands that act via nuclear receptors. The curve of best fit for nonmonotonic concentration response relationships are often inverted U-shaped with effects at intermediate concentrations that are different from effects at higher or lower concentrations. Cytotoxicity is a major mode of action responsible for inverted U-shaped concentration response relationships. However, evidence suggests that ligand selectivity, activation of multiple molecular targets, concerted regulation of multiple opposing endpoints, and multiple ligand binding sites within nuclear receptors also contribute to nonmonotonic concentration response relationships of endocrine active ligands. This review reports the current understanding of mechanisms involved in classical nuclear receptor mediated nonmonotonic concentration response relationships with a focus on studies published between 2012 and 2014." @default.
- W2023786112 created "2016-06-24" @default.
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- W2023786112 date "2014-12-01" @default.
- W2023786112 modified "2023-09-25" @default.
- W2023786112 title "Editorial overview: Endocrine and metabolic diseases: Conversations on endocrine disruptors — rising above the din" @default.
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- W2023786112 doi "https://doi.org/10.1016/j.coph.2014.10.003" @default.
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