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- W2023861938 abstract "A novel series of 1H-indol-1-yl tertiary amine LXR agonists has been designed. Compounds from this series were potent agonists with good rat pharmacokinetic parameters. In addition, the crystal structure of an LXR agonist bound to LXRα will be disclosed." @default.
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- W2023861938 date "2009-02-01" @default.
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- W2023861938 title "Synthesis and SAR of potent LXR agonists containing an indole pharmacophore" @default.
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- W2023861938 doi "https://doi.org/10.1016/j.bmcl.2009.01.004" @default.
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